BDBM392495 N-[2-(4-fluoro-2,3-dimethyl- phenyl)-1H-pyrrolo[2,3- b]pyridin-5-yl]-3,4-dimethyl-1H- pyrazole-5-carboxamide::US10301280, Compound P-2279

SMILES Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(F)c(C)c2C)c1C

InChI Key InChIKey=SCURTBIOSBGLRR-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 392495   

TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM392495(N-[2-(4-fluoro-2,3-dimethyl- phenyl)-1H-pyrrolo[2,...)
Affinity DataKi: <1.00E+3nMAssay Description:The c-kit mutant D816V (or kinase domain thereof) is an active kinase in AlphaScreen. IC50 values are determined with respect to inhibition of c-Kit ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent