BDBM392514 N-(2-methyl-1H-pyrrolo[2,3- b]pyridin-5-yl)-2H-indazole-4- carboxamide::US10301280, Compound P-2301

SMILES Cc1cc2cc(NC(=O)c3cccc4n[nH]cc34)cnc2[nH]1

InChI Key InChIKey=HNBDTSGEWMJFET-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 392514   

TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM392514(N-(2-methyl-1H-pyrrolo[2,3- b]pyridin-5-yl)-2H-ind...)
Affinity DataKi: <1.00E+3nMAssay Description:The c-kit mutant D816V (or kinase domain thereof) is an active kinase in AlphaScreen. IC50 values are determined with respect to inhibition of c-Kit ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent