BDBM393061 5-(3-chloro-4- fluorobenzenesulfon- amidomethyl)-N-(1,3- thiazol-5- ylmethyl)pyrazine-2- carboxamide::US9963434, Table 12.8

SMILES Fc1ccc(cc1Cl)S(=O)(=O)NCc1cnc(cn1)C(=O)NCc1cncs1

InChI Key InChIKey=MYGXBQLPNYBGTO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 393061   

TargetGlutamate receptor ionotropic, NMDA 2A(Homo sapiens (Human))
Luc Therapeutics

US Patent
LigandPNGBDBM393061(5-(3-chloro-4- fluorobenzenesulfon- amidomethyl)-N...)
Affinity DataIC50:  929nMAssay Description:Cell Culture and plating: HEK293 cells expressing NR1/NR2A (Chantest, Cleveland, Ohio) were grown to 70-80% confluency as an adherent monolayer in st...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent