BDBM405071 1-(4-{4-[2-(5-chloro-2- fluorophenyl)acetamido]-1H-1,2,3- triazol-1-yl}butyl)-N-[(5-chloro-2- fluorophenyl)methyl]-1H-1,2,3- triazole-4-carboxamide::US10344025, Example 415::US11370786, Example 415
SMILES Fc1ccc(Cl)cc1CNC(=O)c1cn(CCCCn2cc(NC(=O)Cc3cc(Cl)ccc3F)nn2)nn1
InChI Key InChIKey=DPNMTJJUHYTTJI-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 405071
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Board of Regents, The University of Texas System
US Patent
Board of Regents, The University of Texas System
US Patent
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Board of Regents, The University of Texas System
US Patent
Board of Regents, The University of Texas System
US Patent
Affinity DataIC50: <100nMAssay Description:The inhibition of purified recombinant human GAC by varying concentrations of inhibitors is assessed via a dual-coupled enzymatic assay. The glutamat...More data for this Ligand-Target Pair