BDBM412243 (R)-1'-(4-(2-(3- (fluoromethyl)azetidin- 1-yl)ethoxy)phenyl)- 3',4'-dihydro-1'H- spiro[cyclopentane- 1,2'-naphthalen]-6'-ol::US10399939, Example 122

SMILES Oc1ccc2[C@@H](c3ccc(OCCN4CC(CF)C4)cc3)C3(CCCC3)CCc2c1

InChI Key InChIKey=UTWAZOJGZINIJA-RUZDIDTESA-N

Data  1 EC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 412243   

TargetEstrogen receptor(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM412243((R)-1'-(4-(2-(3- (fluoromethyl)azetidin- 1-yl)etho...)
Affinity DataEC50:  0.451nMAssay Description:The relative efficacies of Formula I compounds as inhibitors of an enzyme activity (or other biological activity) can be established by determining t...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent