BDBM412256 (7S,8R)-8-(4-(2-(3- (fluoromethyl)azetidin- 1-yl)ethoxy)phenyl)- 7-phenyl-5,6,7,8- tetrahydronaphthalen- 1-ol::US10399939, Example 135

SMILES Oc1cccc2CC[C@@H]([C@H](c3ccc(OCCN4CC(CF)C4)cc3)c12)c1ccccc1

InChI Key InChIKey=XWISDJVNQVTQCH-VPUSJEBWSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 412256   

TargetEstrogen receptor(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM412256((7S,8R)-8-(4-(2-(3- (fluoromethyl)azetidin- 1-yl)e...)
Affinity DataEC50:  29.8nMAssay Description:The relative efficacies of Formula I compounds as inhibitors of an enzyme activity (or other biological activity) can be established by determining t...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent