BDBM435239 N-(tert-butyl)-8-((2-(pyridin-3- yl)cyclopropanecarboxamido)methyl)- 5-(3-(trifluoromethoxy)phenyl)-3,4- dihydroisoquinoline-2(1H)- carboxamide (mixture of 4 isomers)::US10568876, Example 4
SMILES CC(C)(C)NC(=O)N1CCc2c(C1)c(CNC(=O)C1CC1c1cccnc1)ccc2-c1cccc(OC(F)(F)F)c1
InChI Key InChIKey=VZVNAVWQXXDDAK-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 435239
Affinity DataIC50: 11.7nMAssay Description:DGAT2 activity was determined by measuring the amount of enzymatic product triolein (1,2,3-Tri(cis-9-octadecenoyl)glycerol) using the membrane prep m...More data for this Ligand-Target Pair