BDBM435262 N-(isoxazol-3-yl)-8-(((trans)-2-(3- methyl-1,2,4-oxadiazol-5- yl)cyclopropanecarboxamido)methyl)- 5-(3-(trifluoromethyl)phenyl)-3,4- dihydroisoquinoline-2(1H)- carboxamide (mixture of 2 isomers)::US10568876, Example 26
SMILES Cc1noc(n1)[C@@H]1C[C@H]1C(=O)NCc1ccc(-c2cccc(c2)C(F)(F)F)c2CCN(Cc12)C(=O)Nc1ccon1
InChI Key InChIKey=ROPGHIKNPSFZDB-FGZHOGPDSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 435262
Affinity DataIC50: 126nMAssay Description:DGAT2 activity was determined by measuring the amount of enzymatic product triolein (1,2,3-Tri(cis-9-octadecenoyl)glycerol) using the membrane prep m...More data for this Ligand-Target Pair