BDBM451398 US10709718, Compound 23

SMILES CC1(C)Oc2ncnc(N)c2N=C1c1ccc(cc1)[C@H]1CC[C@H](CP(O)(=O)C2CC2)CC1

InChI Key InChIKey=QVZDQNCEAFRUNM-WKILWMFISA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 451398   

TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Metabasis Therapeutics

US Patent
LigandPNGBDBM451398(US10709718, Compound 23)
Affinity DataIC50: <10nMAssay Description:The inhibition of DGAT-1 activity can be assessed in intestinal microsome preparations by monitoring the incorporation of radiolabeled fatty acyl-CoA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent