BDBM466938 US10800775, Example 18::isopropyl 4-(1-(2-cyano-1-cyclopentylethyl)-1H-pyrazol-4-yl)- 1H-pyrrolo[2,3-b]pyridine-5-carboxylate, enantiomer 1 single enantiomer, absolute configuration not known
SMILES CC(C)OC(=O)c1cnc2[nH]ccc2c1-c1cnn(c1)[C@H](CC#N)C1CCCC1
InChI Key
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 466938
Affinity DataIC50: <10nMAssay Description:The activity of JAK3 (a.a. 781-1124, ThermoFisher) was quantified by measuring the phosphorylation of SRCtide (FAM-GEEPLYWSFPAKKK-NH2). Kinase reacti...More data for this Ligand-Target Pair