BDBM50009173 CHEMBL3238364

SMILES CCCc1ccc(cc1)N1CC(=O)N(Cc2cc3cnc(nc3n2C)C(=O)N[C@@H](CCCCN)C#N)C1=O

InChI Key InChIKey=TWDYFGPKBAIZRB-FQEVSTJZSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50009173   

TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50009173(CHEMBL3238364)
Affinity DataIC50:  3.30E+5nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-LyspNA (S-2251) peptide as substrate assessed as reduction of enzyme hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50009173(CHEMBL3238364)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human plasma urokinase using Glu-Gly-Arg-pNA (S-2444) peptide as substrate assessed as reduction of enzyme hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50009173(CHEMBL3238364)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human plasma kallikerin using H-D-Phe-Pro-Arg-pNA (S-2302) peptide as substrate assessed as reduction of enzyme hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed