BDBM50009201 CHEMBL3238375

SMILES COc1ccc(Oc2ccc(cc2)N2CC(=O)N(Cc3cc4cnc(nc4n3C)C(=O)N[C@@H](CCCCN)C#N)C2=O)cc1

InChI Key InChIKey=LAMGHZOZXZSKRU-NRFANRHFSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50009201   

TargetPlasminogen(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50009201(CHEMBL3238375)
Affinity DataIC50:  6.40E+4nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-LyspNA (S-2251) peptide as substrate assessed as reduction of enzyme hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50009201(CHEMBL3238375)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of human plasma urokinase using Glu-Gly-Arg-pNA (S-2444) peptide as substrate assessed as reduction of enzyme hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Hiroshima International University

Curated by ChEMBL
LigandPNGBDBM50009201(CHEMBL3238375)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human plasma kallikerin using H-D-Phe-Pro-Arg-pNA (S-2302) peptide as substrate assessed as reduction of enzyme hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed