BDBM50078659 Biphenyl-2-carboxylic acid [5-(5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepine-10-carbonyl)-pyridin-2-yl]-amide::CHEMBL297705

SMILES O=C(Nc1ccc(cn1)C(=O)N1Cc2cccn2Cc2ccccc12)c1ccccc1-c1ccccc1

InChI Key InChIKey=NCQQBBAXLMVSOY-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50078659   

TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078659(Biphenyl-2-carboxylic acid [5-(5H,11H-benzo[e]pyrr...)
Affinity DataIC50:  8.30nMAssay Description:Displacement of P[3H]-AVP from isolated rat kidney medullary V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50078659(Biphenyl-2-carboxylic acid [5-(5H,11H-benzo[e]pyrr...)
Affinity DataIC50:  30nMAssay Description:Displacement of (Phe-3,4,5 [3H]-) AVP from isolated rat hepatic V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed