BDBM50080367 (R)-1-{2-[(Z)-2-(2-Chloro-phenyl)-2-phenyl-vinyloxy]-ethyl}-piperidine-3-carboxylic acid; hydrochloride::CHEMBL540827
SMILES OC(=O)[C@@H]1CCCN(CCO\C=C(\c2ccccc2)c2ccccc2Cl)C1
InChI Key InChIKey=QJFYDLBMZFBGHW-HWLQVLAGSA-N
Data 1 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50080367
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair