BDBM50097567 CHEMBL3588871

SMILES COc1ccc(NC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)NCC2(CCCCC2)c2ccc(OC)cn2)cc1

InChI Key InChIKey=BIVMSUKQESISKU-UHFFFAOYSA-N

Data  8 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50097567   

TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50097567(CHEMBL3588871)
Affinity DataEC50:  430nMAssay Description:Agonist activity at human FPR1 transfected in human HL60 cells assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50097567(CHEMBL3588871)
Affinity DataEC50:  60nMAssay Description:Agonist activity at FPR2 in human PMN assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay in presence of probene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50097567(CHEMBL3588871)
Affinity DataEC50:  96nMAssay Description:Agonist activity at human FPR2 transfected in human HL60 cells assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50097567(CHEMBL3588871)
Affinity DataEC50:  86nMAssay Description:Agonist activity at FPR2 in human neutrophils assessed as induction of calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50097567(CHEMBL3588871)
Affinity DataEC50:  64nMAssay Description:Agonist activity at FPR2 in human PMN assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assay in absence of probenec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50097567(CHEMBL3588871)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human FPR2 expressed in human HL60 cells assessed as induction of calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetfMet-Leu-Phe receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50097567(CHEMBL3588871)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human FPR1 expressed in human HL60 cells assessed as induction of calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50097567(CHEMBL3588871)
Affinity DataEC50:  240nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed