BDBM50098040 2-[1-(2-Bromo-benzyl)-1H-indol-3-yl]-N-isopropyl-N-pyridin-4-ylmethyl-acetamide::CHEMBL168643

SMILES CC(C)N(Cc1ccncc1)C(=O)Cc1cn(Cc2ccccc2Br)c2ccccc12

InChI Key InChIKey=GSQFYOOLDOGGGW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50098040   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50098040(2-[1-(2-Bromo-benzyl)-1H-indol-3-yl]-N-isopropyl-N...)
Affinity DataIC50:  572nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed