BDBM50116243 6-Benzo[1,3]dioxol-5-yl-8-(2-fluoro-benzyl)-3-({[2-(2-fluoro-phenyl)-ethyl]-methyl-amino}-methyl)-2-(4-methoxy-phenyl)-7-methyl-8H-imidazo[1,2-a]pyrimidin-5-one::CHEMBL305034
SMILES COc1ccc(cc1)-c1nc2n(Cc3ccccc3F)c(C)c(-c3ccc4OCOc4c3)c(=O)n2c1CN(C)CCc1ccccc1F
InChI Key InChIKey=YJVWVLHCKCROFB-UHFFFAOYSA-N
Data 1 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50116243
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 67nMAssay Description:Binding evaluated in cloned human Gonadotropin-releasing hormone receptor by displacement of [125 I-Tyr, DLeu, NMeLeu, Pro-NEt]GnRH agonistMore data for this Ligand-Target Pair