BDBM50136534 3-[6-(4-Chloro-phenylsulfanyl)-2-(4-methoxy-phenyl)-3-oxo-2,3-dihydro-pyridazin-4-yl]-N-(2-oxo-azepan-3-yl)-propionamide::CHEMBL138878

SMILES COc1ccc(cc1)-n1nc(Sc2ccc(Cl)cc2)cc(CCC(=O)NC2CCCCNC2=O)c1=O

InChI Key InChIKey=WIQSKJYQQHUGDR-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50136534   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136534(3-[6-(4-Chloro-phenylsulfanyl)-2-(4-methoxy-phenyl...)
Affinity DataIC50:  2.30nMAssay Description:Concentration required to inhibit binding of [125I]NDP-alpha-MSH from membranes prepared from CHO cells expressing human MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed