BDBM50153514 4-{[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl]-hydroxy-methyl}-phenol::CHEMBL186930
SMILES C[C@]12Cc3cnn(c3C=C1CCC[C@@H]2C(O)c1ccc(O)cc1)-c1ccc(F)cc1
InChI Key InChIKey=GEEIYAPDFSGWDJ-KIDMSAQOSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50153514
Affinity DataEC50: 20nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair