BDBM50231050 CHEMBL252013::N-(4-iodophenyl)-4-(trifluoromethoxy)benzamide

SMILES FC(F)(F)Oc1ccc(cc1)C(=O)Nc1ccc(I)cc1

InChI Key InChIKey=IUHUCVXLTXIWPU-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231050   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50231050(CHEMBL252013 | N-(4-iodophenyl)-4-(trifluoromethox...)Copy SMILESCopy InChI

Affinity DataIC50:  280nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI