BDBM50231071 CHEMBL400880::biphenyl-4-carboxylic acid [2-(5-methoxy-1H-indol-3-yl)-ethyl]-amide

SMILES COc1ccc2[nH]cc(CCNC(=O)c3ccc(cc3)-c3ccccc3)c2c1

InChI Key InChIKey=DSZNGEKRTSTCNN-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231071   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50231071(CHEMBL400880 | biphenyl-4-carboxylic acid [2-(5-me...)Copy SMILESCopy InChI

Affinity DataIC50:  370nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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