BDBM50231078 CHEMBL253844::N-(1-(7-methoxynaphthalen-1-yl)propan-2-yl)-4-(trifluoromethoxy)benzamide

SMILES COc1ccc2cccc(CC(C)NC(=O)c3ccc(OC(F)(F)F)cc3)c2c1

InChI Key InChIKey=PUPLVWCDZZBSKT-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231078   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50231078(CHEMBL253844 | N-(1-(7-methoxynaphthalen-1-yl)prop...)Copy SMILESCopy InChI

Affinity DataIC50:  3.10E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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