BDBM50231098 CHEMBL253840::N-(2,3-dihydro-1H-inden-5-yl)-4-(trifluoromethoxy)benzamide

SMILES FC(F)(F)Oc1ccc(cc1)C(=O)Nc1ccc2CCCc2c1

InChI Key InChIKey=IISMKYYEHUKJMC-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231098   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50231098(CHEMBL253840 | N-(2,3-dihydro-1H-inden-5-yl)-4-(tr...)Copy SMILESCopy InChI

Affinity DataIC50:  210nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sid

In DepthDetails ArticlePubMed
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