BDBM50240289 CHEMBL4102586
SMILES Fc1cccc(NS(=O)(=O)c2cc(Cl)c(NCC34CCCN3CCC4)cc2F)n1
InChI Key InChIKey=DGRMYFOOKNVOCV-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50240289
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Department of Discovery Chemistry Merck
Curated by ChEMBL
Department of Discovery Chemistry Merck
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of 50% inactivated human Nav1.5alpha expressed in HEK293 cells at holding potential of -60 mV incubated for 5 mins measured at 10 secs int...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Department of Discovery Chemistry Merck
Curated by ChEMBL
Department of Discovery Chemistry Merck
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of 50% inactivated human Nav1.7alpha expressed in HEK293 cells at holding potential of -60 mV incubated for 5 mins measured at 10 secs int...More data for this Ligand-Target Pair