BDBM50243571 (2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-10-(4-aminobutyl)-4-{[(1S)-1-carbamoyl-2-(naphthalen-2-yl)ethyl]carbamoyl}-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-16-({4-[(methoxycarbamoyl)amino]phenyl}methyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosan-19-yl]-3-(4-chlorophenyl)propanamide::CHEMBL499760

SMILES CONC(=O)Nc1ccc(C[C@@H]2NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc3c[nH]c4ccccc34)NC2=O)[C@@H](C)O)C(=O)N[C@@H](Cc2ccc3ccccc3c2)C(N)=O)NC(=O)[C@H](N)Cc2ccc(Cl)cc2)cc1

InChI Key InChIKey=FAZJEADZIKXOCO-BPBSOZPZSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50243571   

TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50243571((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-10-(4-amin...)
Affinity DataIC50:  313nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst5 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50243571((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-10-(4-amin...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst1 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50243571((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-10-(4-amin...)
Affinity DataIC50:  883nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst4 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50243571((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-10-(4-amin...)
Affinity DataIC50:  157nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst3 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50243571((2R)-2-amino-N-[(4R,7S,10S,13R,16S,19S)-10-(4-amin...)
Affinity DataIC50:  9.30nMAssay Description:Displacement of [125I][LTT]SRIF28 from human cloned sst2 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed