BDBM50256726 CHEMBL4092764

SMILES CCS(=O)(=O)c1ccc(Oc2cccc(NS(=O)(=O)c3ccc(OC)cc3)c2)c(c1)-c1cn(C)c(=O)c2cncn12

InChI Key InChIKey=UMXGEHYOEYQVSN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50256726   

TargetBromodomain-containing protein 4(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50256726(CHEMBL4092764)
Affinity DataIC50:  200nMAssay Description:Inhibition of BRD4-BD2 (333 to 460 residues) (unknown origin) using histone H4 peptide as substrate preincubated for 15 mins followed by addition of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50256726(CHEMBL4092764)
Affinity DataIC50:  140nMAssay Description:Inhibition of BRD4-BD2 (333 to 460 residues) (unknown origin) using histone H4 peptide as substrate preincubated for 15 mins followed by addition of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed