BDBM50257664 (S)-3-amino-N-(3-(N-(3-(3-carbamimidoylphenyl)-1-oxo-1-(piperazin-1-yl)propan-2-yl)sulfamoyl)phenyl)propanamide::CHEMBL493118::US8569313, 54
SMILES NCCC(=O)Nc1cccc(c1)S(=O)(=O)N[C@@H](Cc1cccc(c1)C(N)=N)C(=O)N1CCNCC1
InChI Key InChIKey=IDRHKJAGRANANS-FQEVSTJZSA-N
Data 6 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50257664
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
The Medicines Company (Leipzig)
US Patent
The Medicines Company (Leipzig)
US Patent
Affinity DataKi: 36nMAssay Description:Inhibition assay using matriptase enzymeMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
The Medicines Company (Leipzig)
US Patent
The Medicines Company (Leipzig)
US Patent
Affinity DataKi: 37nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The Medicines Company (Leipzig)
Curated by ChEMBL
The Medicines Company (Leipzig)
Curated by ChEMBL
Affinity DataKi: 880nMAssay Description:Inhibition of uPA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.56E+3nMAssay Description:Inhibition of plasmin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 7.17E+4nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair