BDBM50259808 CHEMBL4093691

SMILES COc1ccc2c(cn(Cc3ccc(cc3)C(=O)NO)c2c1)C(=O)c1cc(OC)c(OC)c(OC)c1

InChI Key InChIKey=VTZNCZMXJPQUPZ-UHFFFAOYSA-N

Data  11 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50259808   

TargetHistone deacetylase 1(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  573nMAssay Description:Inhibition of recombinant human HDAC1 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of recombinant human HDAC2 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  65nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  6.53E+3nMAssay Description:Inhibition of recombinant human HDAC3 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of recombinant human HDAC5 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibition of recombinant human HDAC4 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  1.68E+3nMAssay Description:Inhibition of recombinant human HDAC9 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  651nMAssay Description:Inhibition of recombinant human HDAC11 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  958nMAssay Description:Inhibition of recombinant human HDAC7 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  8.23E+3nMAssay Description:Inhibition of recombinant human HDAC10 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50259808(CHEMBL4093691)
Affinity DataIC50:  390nMAssay Description:Inhibition of recombinant human HDAC8 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed