BDBM50275078 CHEMBL4127542

SMILES OC(=O)CNC(=O)c1ncc(cc1O)-c1cn(Cc2ccc(cc2)C(F)(F)F)nn1

InChI Key InChIKey=ITOHCVOMZJCQTB-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50275078   

TargetEgl nine homolog 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275078(CHEMBL4127542)
Affinity DataIC50:  759nMAssay Description:Inhibition of HIF-PHD2 (181 to 426 residues) (unknown origin) using FITC-HIF1-alpha (556 to 574 residues) as substrate after 60 mins by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed