BDBM50278673 CHEMBL4165366

SMILES OC(=O)CCc1cc(F)c(OCc2c(nsc2C(F)(F)F)-c2ccc(Cl)cc2F)c(F)c1

InChI Key InChIKey=PSUHZRYVUSVFCF-UHFFFAOYSA-N

Data  1 IC50  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50278673   

TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)
Affinity DataEC50:  143nMAssay Description:Agonist activity at PK-tagged human GPR120 long isoform expressed in CHOK1 cells co-expressing EA-tagged beta-arrestin assessed as beta-gal enzyme co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux incubated for 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human GPR40 by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)
Affinity DataEC50:  77nMAssay Description:Agonist activity at mouse GPR120 by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed