BDBM50295950 2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione::CHEMBL541185

SMILES Cn1c2c3ncccc3[nH]c2c(=O)n(C)c1=O

InChI Key InChIKey=DTSCLFDGIVWOGR-UHFFFAOYSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50295950   

TargetAdenosine receptor A3(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50295950(2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene...)
Affinity DataKi:  13.9nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in HEK293T cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50295950(2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene...)
Affinity DataKi:  379nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in HEK293T cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50295950(2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene...)
Affinity DataKi:  893nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2A receptor expressed in HEK293T cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed