BDBM50302304 1,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyridin-2-yl)cyclohexanecarboxamide::CHEMBL568564

SMILES CC1CCCCC1(C)C(=O)Nc1cc(CN2CCOCC2)c(C)cn1

InChI Key InChIKey=XIFPDGUTQDJQGY-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50302304   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302304(1,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302304(1,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]CP55960 from human cloned CB1 receptor after 120 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302304(1,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed