BDBM50323006 1'-(5-(4-chlorophenyl)-4-(2,4-dichlorophenyl)-1-(3-(methylsulfonamido)propyl)-1H-pyrrole-2-carbonyl)-4,4-difluoro-1,4'-bipiperidine-4'-carboxamide::CHEMBL1210782

SMILES CS(=O)(=O)NCCCn1c(cc(c1-c1ccc(Cl)cc1)-c1ccc(Cl)cc1Cl)C(=O)N1CCC(CC1)(N1CCC(F)(F)CC1)C(N)=O

InChI Key InChIKey=YHONTRPKANXJPY-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50323006   

TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50323006(1'-(5-(4-chlorophenyl)-4-(2,4-dichlorophenyl)-1-(3...)
Affinity DataIC50:  1nMAssay Description:Binding affinity to CB1 receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50323006(1'-(5-(4-chlorophenyl)-4-(2,4-dichlorophenyl)-1-(3...)
Affinity DataEC50:  15nMAssay Description:Antagonist activity at CB1 receptor in forskolin-stimulated human U373-MG cells assessed as inhibition of CP-55940-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50323006(1'-(5-(4-chlorophenyl)-4-(2,4-dichlorophenyl)-1-(3...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed