BDBM50334487 4-((3-cyclohexyl-5-(4-(trifluoromethoxy)phenyl)-1H-pyrazol-1-yl)methyl)benzoic acid::CHEMBL1643952

SMILES OC(=O)c1ccc(Cn2nc(cc2-c2ccc(OC(F)(F)F)cc2)C2CCCCC2)cc1

InChI Key InChIKey=YNBPQTVRDVQOFT-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50334487   

TargetGlucagon receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334487(4-((3-cyclohexyl-5-(4-(trifluoromethoxy)phenyl)-1H...)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [125I]glucagon from human GCGR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334487(4-((3-cyclohexyl-5-(4-(trifluoromethoxy)phenyl)-1H...)
Affinity DataIC50:  4.10E+3nMAssay Description:Antagonist activity at human GIPR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed