BDBM50340106 CHEMBL1762824::N-(3-fluoropropyl)-N-(2-methoxyethyl)-8-(2-methoxypyrimidin-5-yl)-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazin-4-amine

SMILES COCCN(CCCF)c1nc(C)nc2c(c(C)nn12)-c1cnc(OC)nc1

InChI Key InChIKey=QIKGXDRLYTUWSV-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50340106   

TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50340106(CHEMBL1762824 | N-(3-fluoropropyl)-N-(2-methoxyeth...)
Affinity DataIC50:  390nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed