BDBM50341294 CHEMBL1766032::N'-(3-Hydroxybenzyl)-aminothiazolo[5,4-b]-N-cyclopropylmethyl-morphinan
SMILES Oc1cccc(CNc2nc3cc4c(C[C@@H]5[C@@H]6CCCC[C@]46CCN5CC4CC4)cc3s2)c1
InChI Key InChIKey=LBJQLPJWKUBKAZ-UTOLSJPLSA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50341294
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.90nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as [35S]GTPgammaS binding by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [3H]Naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation countingMore data for this Ligand-Target Pair