BDBM50346309 CHEMBL1782580::cis-((1S,3R)-3-((3S,4S)-3-hydroxytetrahydro-2H-pyran-4-ylamino)-1-isopropylcyclopentyl)(4-(4-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methanone
SMILES CC(C)[C@@]1(CC[C@H](C1)N[C@H]1CCOC[C@H]1O)C(=O)N1CCN(CC1)c1cc(ccn1)C(F)(F)F
InChI Key InChIKey=PZWALEZJXWWGIX-AWWSKVOZSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50346309
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Displacement of labeled dofetilide from human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 710nMAssay Description:Antagonist activity at human CCR2 by whole blood assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15.4nMAssay Description:Displacement of [125I]MCP1 from human CCR2 preincubated for 30 mins by human whole cell binding assayMore data for this Ligand-Target Pair