BDBM5035 CHEMBL235747::N-(5-tert-Butyl-3,4-dimethyl-1,3-thiazol-2(3H)-ylidene)benzenesulfonamide::N-[(2Z)-5-tert-butyl-3,4-dimethyl-2,3-dihydro-1,3-thiazol-2-ylidene]benzenesulfonamide::thiazolidenebenzenesulfonamide deriv. 10r
SMILES Cc1c(s\c(=N/S(=O)(=O)c2ccccc2)n1C)C(C)(C)C
InChI Key InChIKey=XYRMLZVYRVONRR-PEZBUJJGSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 5035
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical
Yamanouchi Pharmaceutical
Affinity DataIC50: 4.90E+3nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1027,K690N]/[588-1147,K690N](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical
Yamanouchi Pharmaceutical
Affinity DataIC50: >5.00E+4nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgamaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of [3H] CP-55,940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1127,Y768C]/[588-1147,Y768C](Human immunodeficiency virus type 1)
Yamanouchi Pharmaceutical
Yamanouchi Pharmaceutical
Affinity DataIC50: 5.10E+3nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair