BDBM50376253 CHEMBL260464

SMILES CCCCCc1ccc(CC(=O)Nc2cccnc2)cc1

InChI Key InChIKey=VYJQGHFNPZKVTQ-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50376253   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50376253(CHEMBL260464)
Affinity DataKi:  7.26E+3nMAssay Description:Displacement of [3H]RTX from human TRPV1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50376253(CHEMBL260464)
Affinity DataEC50: >5.00E+3nMAssay Description:Activity at human TRPV1 in HEK cells assessed by measuring capsaicin-induced calcium level by FLIPR technologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed