BDBM50395025 CHEMBL2163443::US9708370, CP-1B(i)
SMILES C[C@H](NC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](C)NC(=O)N(Cc1ccc(O)cc1)NC(=O)[C@@H](N)Cc1cnc[nH]1)C(N)=O
InChI Key InChIKey=OZAFXYOETBBYKW-HDSXGYDGSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50395025
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Valorisation-Recherche, Limited Partnership
US Patent
Valorisation-Recherche, Limited Partnership
US Patent
Affinity DataIC50: 7.22E+4nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
TargetEstrogen receptor [D538G](Homo sapiens (Human))
Valorisation-Recherche, Limited Partnership
US Patent
Valorisation-Recherche, Limited Partnership
US Patent
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Valorisation-Recherche, Limited Partnership
US Patent
Valorisation-Recherche, Limited Partnership
US Patent
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair