BDBM50400077 CHEMBL2178403

SMILES O=C(Nc1cccc(c1)C(=O)NCCc1ccncc1)\C=C\Oc1ccc(cc1)C12CC3CC(CC(C3)C1)C2

InChI Key InChIKey=FXQRGQIYHBKGGP-RVDMUPIBSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50400077   

TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Dongguk University-Seoul

Curated by ChEMBL
LigandPNGBDBM50400077(CHEMBL2178403)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of HIF1alpha in human HCT116 cells under hypoxic condition after 16 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed