BDBM50417471 CHEMBL1287953

SMILES CC(C)(C(=O)Nc1ccc(N2CCC3(CCN(CC4CC4)C3)CC2)c(Cl)c1)c1nccc(n1)C(F)(F)F

InChI Key InChIKey=PZAIVSQWZAHADG-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50417471   

TargetNeuropeptide Y-Y2 receptor(Rattus norvegicus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417471(CHEMBL1287953)
Affinity DataKi:  63.1nMAssay Description:Antagonist activity at rat NPY Y2 receptor expressed in HEK cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417471(CHEMBL1287953)
Affinity DataKi:  158nMAssay Description:Antagonist activity at human NPY Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417471(CHEMBL1287953)
Affinity DataKi: >3.98E+3nMAssay Description:Antagonist activity at human NPY Y5 receptor expressed in HEK cells by FLIPR/Ca2+ assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417471(CHEMBL1287953)
Affinity DataKi: >6.31E+3nMAssay Description:Antagonist activity at human NPY Y1 receptor expressed in CHO cells by GTPgammaS35 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed