BDBM50444280 CHEMBL3093641::US9649309, Compound UNC2091A
SMILES CCCCNc1ncc(C(=O)Nc2ccc(cc2)S(=O)(=O)N2CCOCC2)c(N[C@H]2CCNC2)n1
InChI Key InChIKey=PUVADVGBMMQLRI-SFHVURJKSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50444280
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Eshelman School Of Pharmacy�Department Of Pharmacology�Lineberger Compreh
Curated by ChEMBL
Eshelman School Of Pharmacy�Department Of Pharmacology�Lineberger Compreh
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of Mer kinase (unknown origin) using 5-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by microfluidic capillary electrophoresis assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Eshelman School Of Pharmacy�Department Of Pharmacology�Lineberger Compreh
Curated by ChEMBL
Eshelman School Of Pharmacy�Department Of Pharmacology�Lineberger Compreh
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Briefly, activity assays were performed in a 384 well, polypropylene microplate in a final volume of 50 μL of 50 mM Hepes, Ph 7.4 containing 10 ...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Eshelman School Of Pharmacy�Department Of Pharmacology�Lineberger Compreh
Curated by ChEMBL
Eshelman School Of Pharmacy�Department Of Pharmacology�Lineberger Compreh
Curated by ChEMBL
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of Axl kinase (unknown origin) using 5-FAM-KKKKEEIYFFF-CONH2 as substrate after 180 mins by microfluidic capillary electrophoresis assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Eshelman School Of Pharmacy�Department Of Pharmacology�Lineberger Compreh
Curated by ChEMBL
Eshelman School Of Pharmacy�Department Of Pharmacology�Lineberger Compreh
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Tyro-3 kinase (unknown origin) using 5-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by microfluidic capillary electrophoresis as...More data for this Ligand-Target Pair