BDBM50459000 CHEMBL4208543

SMILES Cc1cc2C(=O)NCc2nc1N1CC[C@@H](Oc2ccc3n(C)ncc3c2)[C@@H](F)C1

InChI Key InChIKey=NESYBDNWKKLCGP-QFBILLFUSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50459000   

TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50459000(CHEMBL4208543)
Affinity DataEC50:  17nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine receptor M4 expressed in CHO-K1 cells coexpressing Galphaqi5 assessed as increase in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed