BDBM50475035 CHEMBL362804::TP-109

SMILES COc1ccc(C[C@H](NC(=O)Cc2cccc3ccccc23)C(=O)N[C@@H](C(C)C)C(=O)NC(Cc2ccc(O)cc2)C=O)cc1

InChI Key InChIKey=ROOOPKPTTPSQLF-CJIPUWSSSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50475035   

LigandPNGBDBM50475035(CHEMBL362804 | TP-109)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475035(CHEMBL362804 | TP-109)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475035(CHEMBL362804 | TP-109)
Affinity DataIC50:  20nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed