BDBM50500410 CHEMBL3745799
SMILES Fc1ccc(cc1)-c1cn(nn1)[C@@H]1CN2CCC1CC2
InChI Key InChIKey=AGNZBWKVIGAWTQ-OAHLLOKOSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50500410
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
Mahidol University
Curated by ChEMBL
Mahidol University
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]epibatidine from human alpha3beta4 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universite Orleans
Curated by ChEMBL
Universite Orleans
Curated by ChEMBL
Affinity DataKi: 114nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAchR in rat frontal corticesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Mahidol University
Curated by ChEMBL
Mahidol University
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Displacement of [3H]MLA from human alpha7 nAChR transfected in human SH-SY5Y cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Mahidol University
Curated by ChEMBL
Mahidol University
Curated by ChEMBL
Affinity DataKi: 515nMAssay Description:Displacement of [3H]epibatidine from human alpha4beta2 nAChR transfected in HEK293 cell membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair