BDBM50512954 CHEMBL4527339
SMILES CN1C[C@@H](C[C@@H](C1)c1ccc(Cl)c(c1)C(F)(F)F)Nc1nc2cc[nH]c2c(=O)n1C
InChI Key InChIKey=POPPPIOICRXWNP-QWHCGFSZSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50512954
Affinity DataKd: 138nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of biotinylated peptide binding to human GST-tagged PCAF bromodomain expressed in Escherichia coli Rosetta (DE3) measured after 15 hrs by ...More data for this Ligand-Target Pair