BDBM50546051 CHEMBL4798497

SMILES COc1cc(N2CC(C2)NC(=O)c2sc3nnc(Cl)c(C)c3c2N)c(Cl)cn1

InChI Key InChIKey=KQHAXBIOQNUZKY-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50546051   

TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Vanderbilt University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546051(CHEMBL4798497)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of human M2 receptor/Gqi5 in presence of EC20 glutamate by calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50546051(CHEMBL4798497)
Affinity DataEC50:  10nMAssay Description:Positive allosteric modulation of human M4 receptor/Gqi5 in presence of EC20 glutamate by calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed