BDBM50547126 CHEMBL4763473

SMILES FC(F)(F)c1cccc(Nc2ccccc2C(=O)CCl)c1

InChI Key InChIKey=JPVDFGYNLUBCSD-UHFFFAOYSA-N

Data  1 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50547126   

TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547126(CHEMBL4763473)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547126(CHEMBL4763473)
Affinity DataIC50:  1.41E+4nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Max Planck Institute Of Molecular Physiology

Curated by ChEMBL
LigandPNGBDBM50547126(CHEMBL4763473)
Affinity DataIC50:  800nMAssay Description:Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed