BDBM50582526 CHEMBL5089555
SMILES Cc1ccc(NC(=O)COc2ccc3cc(\C=C4\SC(=O)NC4=O)ccc3c2)cc1
InChI Key InChIKey=SZXUDKIXIBVQCU-RGVLZGJSSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50582526
TargetHistone deacetylase 4(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataEC50: 1.22E+3nMAssay Description:Partial agonist activity at Gal4-fused human PPARgamma LBD in HepG2 cells assessed as transactivation incubated for 20 hrs measured by luminometerMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Bharati Vidyapeeth'S College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair